Tesofensine, single vial

Triple monoamine reuptake inhibitor

Tesofensine

NOT A PEPTIDE — small molecule. A bicyclic azabicyclo-octane compound, not a chain of amino acids.. Supplied for laboratory research use only.

  • Small molecule (monoamine reuptake inhibitor) -- not a peptide
  • Not approved; own Phase 2 showed cardiovascular safety signal
  • Combination product Tesomet approved in Mexico only
  • Supplied for laboratory research use only. Not for human or veterinary use.
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Research use only. Not for human or veterinary use or consumption. This product is not approved by the FDA and is not intended to diagnose, treat, cure or prevent any disease.

What it is
CompoundTesofensine
ClassTriple monoamine reuptake inhibitor
CompositionNOT A PEPTIDE — small molecule. A bicyclic azabicyclo-octane compound, not a chain of amino acids.
FormCapsules or raw powder, supplied in a vial
OriginatorNeuroSearch, originator; later developed by Saniona
Development status

Tesofensine is not approved by the FDA for any indication.

Development status is stated above. No efficacy claim is made on this page.

Shipping & returns
ReturnsNinety days from delivery. Contact us and we will refund the purchase price.
Tesofensine $239.99

The specifics

The details, if you want them.

ClassTriple monoamine reuptake inhibitor
Molecule typeSmall molecule — not a peptide
Regulatory historyUS development stalled after a cardiovascular safety signal in its own Phase 2 trial
FormRaw powder or capsule (not a reconstituted vial)
Receptor target(s)Serotonin transporter, noradrenaline transporter, dopamine transporter

Development

Where it is up to.

Its own Phase 2 trial identified a cardiovascular safety signal that halted US development; that signal remains unresolved. No later-phase US data exists.

Questions

The questions people actually ask.

What is tesofensine?
A small molecule, not a peptide, that inhibits reuptake of three neurotransmitters — serotonin, noradrenaline, and dopamine.
Is tesofensine actually a peptide?
No. It's a small molecule with no amino-acid sequence, despite sometimes appearing in peptide catalogues. Describing it as a peptide is inaccurate.
Is tesofensine approved by the FDA?
No. US development stalled after an unresolved cardiovascular safety signal in its own Phase 2 trial. A combination product is approved only in Mexico.
What does "Research Use Only" mean?
Research Use Only means exactly that: intended for laboratory and research settings only, not for human or animal use, consumption, diagnosis, treatment, cure, or prevention of any disease.
What is your refund policy?
Ninety days from delivery. If you decide against it inside that window, contact hello@getmrpeps.com and we will refund the purchase price. Damaged or incorrect orders are replaced or refunded regardless.